I-Enrofloxacin liyeza elibulala iintsholongwane elibanzi kwizilwanyana ezikudidi lwe-flurofenolone. I-Escherichia coli, i-Salmonella, i-Klebsiella, i-Brucella, i-Pasteurella, i-Actinobacillus pleuropneumoniae, i-Erysipelas, i-Proteus, i-Serratia marcescens, i-Corynebacterium pyogenes, i-Portella septicarum Inefuthe elihle kwiibhaktheriya, i-Staphylococcus aureus, i-mycoplasma, i-chlamydia, njl.njl., kodwa inefuthe elibuthathaka kwi-Pseudomonas aeruginosa kunye ne-Streptococcus kwaye inefuthe elibuthathaka kwiibhaktheriya ezingena-anaerobic. Inefuthe elicacileyo le-antibacterial post-effect kwiibhaktheriya ezinobuthathaka.
Le mveliso ifunxwa ngokukhawuleza nangokupheleleyo ngenaliti ye-intramuscular. Ukufumaneka kwayo yi-91.9% kwiihagu kunye ne-82% kwiinkomo zobisi. Isasazeka kakhulu kwizilwanyana kwaye ingangena ngokulula kwizicubu kunye nolwelo lomzimba. Ngaphandle kolwelo lwe-cerebrospinal, uxinaniso lwamayeza phantse kwizicubu luphezulu kunolo lusegazini. I-Pulp. I-metabolism yesibindi ibandakanya kakhulu ukususwa kweqela le-ethyl yeringi ye-7-crosin ukuvelisa i-ciprofloxacin, kulandele i-oxidation kunye ne-glucuronic acid conjugation, ikakhulu ikhutshwa ngezintso (ngokukhutshwa kwetyhubhu yezintso kunye nokuhluzwa kwe-glomerular), i-15% ukuya kwi-50% Ikhutshwa ingatshintshanga kumchamo. Isusa isiqingatha Ubomi bomzimba buyahluka kakhulu kwiintlobo ezahlukeneyo zezilwanyana kunye neendlela ezahlukeneyo zokusetyenziswa. Ukususwa kwesiqingatha sobomi emva kokufakwa kwe-intramuscular.
ukusebenzisana kwamayeza: (1) Le mveliso inefuthe lokusebenzisana xa idityaniswe nee-amino sugar okanye i-penicillin ye-wide-spectrum. (2) Ii-ion zesinyithi ezinzima ezifana ne-Ca2+, i-Mg2+, i-Fe; kunye ne-Al Children zinokusebenzisana nale mveliso kwaye zichaphazele ukufunxwa. (3) Xa zisetyenziswa kunye ne-theophylline kunye ne-caffeine, izinga lokubopha iiproteni ze-plasma linokuncipha, uxinzelelo lwe-theophylline kunye ne-caffeine egazini luya kwanda ngendlela engaqhelekanga, kwaye neempawu zetyhefu ye-theophylline zinokubakho. (4) Le mveliso inefuthe lokuthintela ii-enzymes zamayeza esibindi kwaye inokunciphisa izinga lokususwa kwamayeza axutywa kakhulu esibindini.
Umsebenzi kunye nokusetyenziswa: Ii-antibiotics zeFlufenolone. Zisetyenziselwa izifo zeebhaktheriya kunye nosulelo lwe-mycoplasma kwimfuyo nakwiinkukhu.
Ixesha leposi: Epreli-26-2024 | 1 imbono


