I-Albendazole yi-anthelmintic yokwenziwa ekwiqela le-benzimidazole-derivatives enomsebenzi ngokuchasene neentlobo ngeentlobo zeempethu kwaye kwinqanaba eliphezulu ledosi ikwachasene nezigaba ze-liver fluke zabantu abadala.
I-Albendazole idityaniswe neproteni ye-microtubule ye-eelworm kwaye idlala indima. Emva kokuba i-albenzene idityaniswe ne-β-tubulin, inokuthintela ukungalingani phakathi kwe-albenzene kunye ne-α tubulin edibana ibe yi-microtubules. Ii-Microtubules zezona zakhiwo zisisiseko zeeyunithi ezininzi zeeseli. Ubudlelwane be-Albendazole ne-nematodes tubulin buphezulu kakhulu kunobudlelwane be-tubulin yezilwanyana ezincancisayo, ngoko ke ubuthi kwizilwanyana ezincancisayo buncinci.
Ukuthintela nonyango lwezifo zeentshulube kumathole nakwiinkomo ezifana nezi:
Iimpethu zesisu:IBunostomum, Cooperia, Chabertia, Haemonchus, Nematodirus, Oesophagostomum, Ostertagia, Strongyloides kunye neTrichostrongylus spp.
Iimpethu zemiphunga:I-Dictyocaulus viviparus kunye ne-D. filaria.
Iimpethu ezirhabaxa:I-Monieza spp.
I-Liver-fluke:umntu omdala one-Fasciola hepatica.
I-Albendazole ikwanomphumo wokubulala iintsholongwane.
Ukunikezelwa kweyeza kwiintsuku zokuqala ezingama-45 zokukhulelwa.
Iimpendulo ze-Hypersensitivity.
Ukulawulwa ngomlomo.
Kwiintshulube ezingqukuva, ii-tapeworms:
Iinkomo / inyathi / ihashe / igusha / ibhokhwe: 5mg/kg ubunzima bomzimba
Inja/ikati: 10 ukuya kwi-25mg/kg ubunzima bomzimba
Ngee-flukes:
Iinkomo/iinyathi: 10mg/kg ubunzima bomzimba
Igusha/ibhokhwe: 7.5mg/kg ubunzima bomzimba
Amathole neenkomo: 1 bolus kwi 300 kg nganye. ubunzima bomzimba.
Kwi-liver-fluke:
I-bolus e-1 kwi-250 kg nganye. ubunzima bomzimba.
Gcina kude nokufikelela kwabantwana.
Iminyaka emi-3.
- Ngenyama:Iintsuku ezili-12.
- Ngobisi:Iintsuku ezi-4.
Gcina kwindawo epholileyo neyomileyo ekhuselweyo ekukhanyeni.